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            ApexBio B7718說明書

             更新時間:2018-08-16 點(diǎn)擊量:1769

            ApexBio是生物研究用肽和實(shí)驗(yàn)室試劑的主要供應(yīng)商。我們在細(xì)胞凋亡,表觀遺傳學(xué),癌癥生物學(xué)等研究領(lǐng)域擁有廣泛的產(chǎn)品線。Apexbio還提供定制服務(wù),包括肽合成,抗體生產(chǎn)和分析開發(fā)。

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            (R)-PFI 2 hydrochloride 
            SETD7 histone lysine methyltransferase inhibitor

            窗體頂端

            Catalog No.B7718

            (R)-PFI 2鹽酸鹽 
            SETD7組蛋白賴氨酸甲基轉(zhuǎn)移酶抑制劑

            窗體底端

            Size

            Price

            10mg

            $302.00

             

            化學(xué)性質(zhì)

            卡號

            1627607-87-7

            SDF

            下載SDF

            化學(xué)名稱

            (R)-8-氟-N-(1-氧代-1-(吡咯烷-1-基)-3-(3-(san氟甲基)苯基)丙-2-基)-1,2,3,4-四氫異喹啉-6-磺酰胺鹽酸鹽

            Canonical SMILES

            FC1 = C2CNCCC2 = CC(S(N [ C ]](C(N3CCCC3)= O)([H])CC4 = CC(C(F)(F)F)= CC = C4)(= O)= O )= C1.Cl

            23 H 25 F 4 N 3 O 3 S.HCl

            M.Wt

            535.98

            可溶性

            溶于DMSO> 10 mM

            存儲

            儲存在-20°C

            物理外觀

            結(jié)晶固體

            運(yùn)輸條件

            評估樣品解決方案:裝有藍(lán)色冰。所有其他可用尺寸:根據(jù)要求提供RT或藍(lán)冰

            一般提示

            為了獲得更高的溶解度,請在37℃下加熱管并在超聲波浴中搖動一段時間。庫存溶液可在-20℃以下儲存數(shù)月。

             

             

             

            1. Cat.No                 .Product                                      NameInformation
            2. A8181                   (-)-JQ1BET                               bromodomain inhibitor
            3. B7679                 (R)-(+)-Etomoxir sodium salt            carnitine palmitoyltransferase I (CPT1) inhibitor
            4. B7718               (R)-PFI 2 hydrochloride                     SETD7 histone lysine methyltransferase inhibitor
            5. C4834                   (S)-PFI-2 (hydrochloride)             Negative control of (R)-PFI 2 hydrochloride
            6. A4510               1,2,3,4,5,6-HexabromocyclohexaneJ          AK2 tyrosine kinase inhibitor
            7. C4119              2',3',5'-triacetyl-5-Azacytidine   prodrug form of 5-azacytidine, a DNA methyltransferase inhibitor
            8. B5972               2,4-Pyridinedicarboxylic Acid                 Histone LSD inhibitor
            9. C4445                      2-D08                               Sumoylation inhibitor
            10. B5969                2-hexyl-4-Pentynoic Acid                 Potent and robust HDACs inhibitor
            11. A4188                  2-Methoxyestradiol (2-MeOE2)        Apoptotic, antiproliferative and antiangiogenic agen
            1. A8182         3-Deazaneplanocin A (DZNep) hydrochloride      SAHH and ENZ2 inhibitor
            2. A1905        3-Deazaneplanocin,DZNep             S-adenosylhomocysteine and EZH2 inhibitor
            3. C3552        4'-bromo-Resveratrol                        Sirt1 and Sirt3 inhibitor
            4. A4524         4-HQN                                       PARP inhibitor
            5. C4018         4-iodo-SAHA         class I and class II histone deacetylase (HDAC) inhibitor
            6. B4106       4SC-202                                  Class I HDAC inhibitor
            7. C3505       5-(N,N-dimethyl)-Amiloride (hydrochloride)      NHE1, NHE2, and NHE3 inhibitor
            8. A1907         5-Azacytidine                           DNA methyltransferase inhibitor.
            9. B4947        A 366                      G9a/GLP histone lysine methyltransferase inhibitor
            10. A4160        A-966492                                PARP-1/-2 inhibitor, highly potent
            1. B1182           ABC294640                           Sphingosine kinase 2 inhibitor,selective and competitive
            2. A3002         ABT-888 (Veliparib)                                      Potent PARP inhibitor
            3. B5936           ACY-241                                Selective and orally active HDAC6 inhibitor
            4. B6120          Adox                                          indirect methyltransferase inhibitor
            5. A4158         AG-14361                                     Potent PARP1 inhibitor
            6. B7323            AGK 2                                        SIRT2 inhibitor, potent and selective
            7. C5709               AGK7                                     cell-permeable, selective inhibitor of SIRT2
            8. B4713              AK-7                                   selective and brain-permeable SIRT2 inhibitor
            9. A4542            Alexidine dihydrochloride                                PTPMT1 inhibitor
            10. A4119               AMG-900                                           Aurora kinase inhibitor

             

             

             

            上海起發(fā)實(shí)驗(yàn)試劑有限公司是實(shí)驗(yàn)試劑一站式采購服務(wù)商

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            2:產(chǎn)品種類齊全,經(jīng)營超過700多品牌,基本涵蓋所有生物實(shí)驗(yàn)試劑耗材。

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            4:富有競爭力的價格優(yōu)勢,絕大部分價格有優(yōu)勢。

            5:多年積累良好的信譽(yù),大部分客戶提供貨到付款服務(wù)??蛻舭ㄇ迦A、北大、交大、復(fù)旦、中山等100多所高校,ROCHE,阿斯利康、國藥、fisher等知藥企。

            6:我們還是Santa,Advanced Biotechnologies Inc,Athens Research & Technology,bangs,BBInternational,crystalchem,dianova,FD Neurotechnologies,Inc. FormuMax Scientific,Inc, Genebridege, Glycotope Biotechnology GmbH; iduron,Innovative Research of America, Ludger, neuroprobe,omicronbio, Polysciences,prospecbi, QA-BIO,quickzyme,RESEARCH DIETS,INC,sterlitech;sysy,TriLink BioTechnologies,Inc;worthington-biochem,zyagen等幾十家國外公司授權(quán)代理。

            7:我們還是invitrogen,qiagen,MiraiBioam,sigma;neb,roche,merck, rnd,BD, GE,pierce,BioLegend等知*批發(fā),歡迎合作。

             

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